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中文名称:
SEN 12333
英文名称:
SEN 12333
CAS No.:
874450-44-9
分子式:
C₂₀H₂₅N₃O₂
分子量:
339.43
技术问答
游客JZ2108199770
2021-08-19 09:09
问 SEN 12333用途是什么?
描述:SEN 12333是做什么用的?哪里可以用到SEN 12333?
答
SEN 12333 is a nicotinic acetylcholine receptor (nAChR) agonist. SEN 12333 displays functional antagonism at histamine H3 receptors (IC50 = 103 nM) and weak agonist activity at human ganglionic α3 nAC
hRs (IC50 = 8.5 渭M). Neuroprotective in a rodent model of quisqualic acid-induced cholinergic degeneration. SEN 12333 is a brain penetrant and orally bioavailable.
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Tags:SEN 12333,874450-44-9,cas号:874450-44-9,cas:874450-44-9
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